Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM452570'
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech, Inc.

US Patent
LigandPNGBDBM452570(3-((3-((3R,5R)-5-(4- chlorophenyl)tetra- hydrofura...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:The IC50 (effective concentration) of compounds on the human TRPA1 channel was determined using a FLIPR Tetra instrument. CHO cells expressing TRPA1 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q251429WUS Patent
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech, Inc.

US Patent
LigandPNGBDBM452570(3-((3-((3R,5R)-5-(4- chlorophenyl)tetra- hydrofura...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:The IC50 (effective concentration) of compounds on the human TRPA1 channel was determined using a FLIPR Tetra instrument. CHO cells expressing TRPA1 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q251429WUS Patent