Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM50022349'
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50022349(CHEMBL3299024)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human TRPA1 expressed in CHO-TREX cells assessed as inhibition of cinnamaldehyde-induced calcium flux incubated 10 mins prior ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TKTPubMed
TargetTransient receptor potential cation channel subfamily A member 1(Mus musculus)
Genomics Institute of the Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50022349(CHEMBL3299024)copy SMILEScopy InChI
Affinity DataIC50: 254nMAssay Description:Antagonist activity at mouse TRPA1 expressed in CHO-TREX cells assessed as inhibition of cinnamaldehyde-induced calcium flux incubated 10 mins prior ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TKTPubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Genomics Institute of the Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50022349(CHEMBL3299024)copy SMILEScopy InChI
Affinity DataIC50: 627nMAssay Description:Antagonist activity at rat TRPA1 expressed in CHO-TREX cells assessed as inhibition of cinnamaldehyde-induced calcium flux incubated 10 mins prior to...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TKTPubMed