BindingDB PrimarySearch

Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM50263524'

Transient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))TBA

BDBM50263524(CHEMBL4096004 | US11236046, Example 4)copy SMILEScopy InChI

IC50: 819nMAssay Description:IC50s (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells expressing...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Details
BindingDB Entry DOI: 10.7270/Q25T3PPTUS Patent

Transient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))TBA

BDBM50263524(CHEMBL4096004 | US11236046, Example 4)copy SMILEScopy InChI

IC50: 4.40E+3nMAssay Description:Inhibition of human TRPA1 expressed in HEK293 cells assessed as inhibition of cinnamaldehyde-induced Ca2+ influx preincubated for 20 mins followed by...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2VX0JZVPubMed