Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM50263527'
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Pharmaron-Beijing Co. Ltd. , 6 Taihe Road, BDA , Beijing 100176 , P. R. China.

Curated by ChEMBL
LigandPNGBDBM50263527(CHEMBL4087767)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human TRPA1 expressed in HEK293 cells assessed as inhibition of cinnamaldehyde-induced Ca2+ influx preincubated for 20 mins followed by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0JZVPubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Pharmaron-Beijing Co. Ltd. , 6 Taihe Road, BDA , Beijing 100176 , P. R. China.

Curated by ChEMBL
LigandPNGBDBM50263527(CHEMBL4087767)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human TRPA1 expressed in CHO cells measured by calcium based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9FKVPubMed
LigandPNGBDBM50263527(CHEMBL4087767)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Antagonist activity at rat TRPA1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9FKVPubMed