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TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Kissei Pharmaceutical Co., Ltd.
Curated by ChEMBL
Kissei Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Antagonist activity at human recombinant TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium increase by Fluo-4 AM base...More data for this Ligand-Target Pair
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