Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50331285'
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Renovis, Inc.

Curated by ChEMBL
LigandPNGBDBM50331285(2-(5-(benzyloxy)-2-methyl-1H-indol-3-yl)ethanamine...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human TRPM8 receptor expressed in human T-REx-293 cells assessed as inhibition of menthol-induced 45calcium influx treated 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN459HPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Renovis, Inc.

Curated by ChEMBL
LigandPNGBDBM50331285(2-(5-(benzyloxy)-2-methyl-1H-indol-3-yl)ethanamine...)copy SMILEScopy InChI
Affinity DataIC50: 2.36E+3nMAssay Description:Antagonist activity at human TRPM8 receptor expressed in human T-REx-293 cells assessed as inhibition of icilin-induced 45calcium influx treated 5 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN459HPubMed