Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50512055'
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition in WS5-induced increase in calcium influx incubated for 10 mins p...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University of Hull
Curated by ChEMBL
University of Hull
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition in WS5-induced increase in calcium influx incubated for 10 mins p...More data for this Ligand-Target Pair