Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50544531' TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University of Salerno
Curated by ChEMBL
University of Salerno
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK-293/TRPM8 exon1 K3 cells assessed as inhibition of menthol-induced current response by whole-cell...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno
Curated by ChEMBL
University of Salerno
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium flux preincubated for 60 mins followed b...More data for this Ligand-Target Pair
