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TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Neurogen Corporation
Curated by ChEMBL
Neurogen Corporation
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Neurogen Corporation
Curated by ChEMBL
Neurogen Corporation
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Neurogen Corporation
Curated by ChEMBL
Neurogen Corporation
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human TRPV1 receptorMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Neurogen Corporation
Curated by ChEMBL
Neurogen Corporation
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:In vitro antagonistic activity on VR1 receptor in [Ca2+] influx assay in rat dorsal root ganglionMore data for this Ligand-Target Pair
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