Found 1 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 4' and Ligand = 'BDBM230252' TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
SHIONOGI & CO., LTD.
US Patent
SHIONOGI & CO., LTD.
US Patent
Affinity DataKi: 130nM ΔG°: -40.9kJ/mole IC50: 420nMT: 2°CAssay Description:Test Example 1: (1) The TRPV4 inhibitory activity was measured using CHO-K1 cells stably expressing human TRPV4 (hTRPV4/CHO cells). (2) In the day be...More data for this Ligand-Target Pair
