Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 4' and Ligand = 'BDBM50117640'
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Renovis, Inc.

Curated by ChEMBL
LigandPNGBDBM50117640(CHEMBL3613639)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1THPPubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
Renovis, Inc.

Curated by ChEMBL
LigandPNGBDBM50117640(CHEMBL3613639)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1THPPubMed