Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Transitional endoplasmic reticulum ATPase' and Ligand = 'BDBM50562860'
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562860(CHEMBL4762311)copy SMILES
Affinity DataIC50: 600nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562860(CHEMBL4762311)copy SMILES
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562860(CHEMBL4762311)copy SMILES
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of His6-tagged p97 C522A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed