Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor' and Ligand = 'BDBM82258'
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6T7VPubMed
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]-AII from the Angiotensin II receptor isolated from the liver of ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9DHJPubMed
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Competitive inhibition of Angiotensin II receptor binding of radiolabeled AII to rat adrenal glomerulosa tissue by 50%More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Z03B9M
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of radioligand [3H]angiotensin II binding to angiotensin II receptor of rat adrenal cortical membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QN690PPubMed
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN98BK