Compile Data Set for Download or QSAR
Found 12 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor B' and Ligand = 'BDBM50009714'
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DR2TJSPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Binding affinity against angiotensin II receptor type 1 (AT1) from rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28W3CCPPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X28DXPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 8.20nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2W4J
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 measured by ability to displace [125I]- A II from its specific binding site in rat liver membran...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22Z14M0PubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Concentration of the compound required to inhibit binding of radioligand [125I]-AII to angiotensin II receptor, type 1 in rat adrenal glomerulosa tis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930S4RPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro antagonistic activity by displacement of [125I]-Sar1-Ile8-A II at the rat adrenal cortical aorta Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55MKHPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7MRPPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98746PubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of [125I]-angiotensin-II binding to the angiotensin II receptor type 1 in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53JXMPubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125-I]-labeled angiotensin II binding to AT1 receptor in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94VB
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+4nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0MDWPubMed