Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM181017'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
PHARMACYCLICS, INC.

US Patent
LigandPNGBDBM181017(US9133201, 6)copy SMILEScopy InChI
Affinity DataIC50: 0.520nMpH: 7.4Assay Description:Btk kinase activity was determined using a time-resolved fluorescence resonance energy transfer (TR-FRET) methodology. Measurements were performed in...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ02KCUS Patent