Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM230105'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM230105(US10106559, Example 29 | US10435415, Example 29 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMpH: 7.4 T: 2°CAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), ATP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BK1B6SUS Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM230105(US10106559, Example 29 | US10435415, Example 29 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53P6VUS Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM230105(US10106559, Example 29 | US10435415, Example 29 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R2CUS Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM230105(US10106559, Example 29 | US10435415, Example 29 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMpH: 7.4 T: 2°CAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SF2Z7QUS Patent