Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM377360'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Curacyte Chemistry GmbH

LigandPNGBDBM377360(US10266491, Example 28 | US10676434, Example 28 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112M3US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Curacyte Chemistry GmbH

LigandPNGBDBM377360(US10266491, Example 28 | US10676434, Example 28 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 ATP (20 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HT2SG3US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Curacyte Chemistry GmbH

LigandPNGBDBM377360(US10266491, Example 28 | US10676434, Example 28 | ...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CN76Z8US Patent