Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM377487'
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Curacyte Chemistry GmbH

LigandPNGBDBM377487(4-(1-acryloylindolin-6-yl)-3- fluoro-7-(2-hydroxye...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112M3US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Curacyte Chemistry GmbH

LigandPNGBDBM377487(4-(1-acryloylindolin-6-yl)-3- fluoro-7-(2-hydroxye...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 ATP (20 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HT2SG3US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Curacyte Chemistry GmbH

LigandPNGBDBM377487(4-(1-acryloylindolin-6-yl)-3- fluoro-7-(2-hydroxye...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:To V-bottom 384-well plates were added test compounds, human recombinant Btk (1 nM, Invitrogen Corporation), fluoresceinated peptide (1.5 μM), A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CN76Z8US Patent