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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK [386-659]' and Ligand = 'BDBM467396'
Target
Tyrosine-protein kinase BTK [386-659]
(Homo sapiens (Human))
Janssen Pharmaceutica NV
US Patent
Ligand
BDBM467396
((R,E)-N-(1-(2-Cyano-3-cyclopropylacryloyl)piperidi...)
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Affinity Data
IC50: 10nM
Assay Description:
A BTK kinase lanthascreen binding assay monitors compound binding to unphosphorylated-BTK kinase domain (UP-BTK), by competing with a fluorescent lab...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q22V2K6B
US Patent