Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK [C481S]' and Ligand = 'BDBM499811'
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
ArQule, Inc.

US Patent
LigandPNGBDBM499811(US11020398, Compound I-123 | US20230364079, Exampl...)copy SMILES
Affinity DataIC50: 0.390nMAssay Description:Enzyme assay using full length recombinant active form of wild-type BTK and BTK-C481S was measured as described previously (Anastassiadis T, et al., ...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
ArQule, Inc.

US Patent
LigandPNGBDBM499811(US11020398, Compound I-123 | US20230364079, Exampl...)copy SMILES