Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK [357-620,Y512E]' and Ligand = 'BDBM213219'
TargetTyrosine-protein kinase ITK/TSK [357-620,Y512E](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM213219((S)-1-(3-((4-(Morpholinomethyl)-6-(thiazolo[5,4-b]...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:This assay is based on the binding and displacement of Alexa-fluor 647-labeled ATP-competitive kinase inhibitor tracer 236. Binding of the tracer is ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1JSKPubMed
TargetTyrosine-protein kinase ITK/TSK [357-620,Y512E](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM213219((S)-1-(3-((4-(Morpholinomethyl)-6-(thiazolo[5,4-b]...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:This assay is based on the binding and displacement of Alexa-fluor 647-labeled ATP-competitive kinase inhibitor tracer 236. Binding of the tracer is ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1JSKPubMed