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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK [357-620,Y512E]' and Ligand = 'BDBM213221'
Target
Tyrosine-protein kinase ITK/TSK [357-620,Y512E]
(Homo sapiens (Human))
GlaxoSmithKline
Ligand
BDBM213221
((S)-1-(3-((4-(Piperidin-1-ylmethyl)-6-(thiazolo[5,...)
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Affinity Data
IC50: 6.30nM
Assay Description:
This assay is based on the binding and displacement of Alexa-fluor 647-labeled ATP-competitive kinase inhibitor tracer 236. Binding of the tracer is ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2ZW1JSK
PubMed