Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK [357-620,Y512E]' and Ligand = 'BDBM213223'
Target
Tyrosine-protein kinase ITK/TSK [357-620,Y512E]
(Homo sapiens (Human))
GlaxoSmithKline
Ligand
BDBM213223
(1-((S)-3-((4-((((R)-3,3-Dimethylbutan-2-yl)amino)m...)
copy SMILES
copy InChI
Affinity Data
IC50: 7.90nM
Assay Description:
This assay is based on the binding and displacement of Alexa-fluor 647-labeled ATP-competitive kinase inhibitor tracer 236. Binding of the tracer is ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2ZW1JSK
PubMed