Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK1' and Ligand = 'BDBM50274583'
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Eberhard Karls University T£bingen

Curated by ChEMBL
LigandPNGBDBM50274583(CHEMBL4125861)copy SMILEScopy InChI
Affinity DataIC50: 117nMAssay Description:Inhibition of human JAK1 using poly[Glu:Tyr] (4:1) as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6988PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Eberhard Karls University T£bingen

Curated by ChEMBL
LigandPNGBDBM50274583(CHEMBL4125861)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of kinase tracer-04 binding to C-terminal NanoLuc tagged full length JAK1 (unknown origin) expressed in HEK cells by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6988PubMed