TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 578nMAssay Description:Inhibition of human JAK2 using poly[Glu:Tyr] (4:1) as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 2.55E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay affinity-purified GST fusions of the active kinase domains (GST-Jak1(866-1154), GST-Jak2(808-1132), GST-Jak3(811-1124) and GST-Tyk2(888-...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibition of GST-tagged Jak2 expressed in insect cells using 20 uM ATPMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
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