Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK3' and Ligand = 'BDBM50274605'
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen

Curated by ChEMBL
LigandPNGBDBM50274605(CHEMBL4128266)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen

Curated by ChEMBL
LigandPNGBDBM50274605(CHEMBL4128266)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human JAK3 (781 to 1124 residues) expressed in baculovirus expression system assessed as reduction in polypeptide substrate...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen

Curated by ChEMBL
LigandPNGBDBM50274605(CHEMBL4128266)copy SMILEScopy InChI
Affinity DataEC50:  740nMAssay Description:Inhibition of kinase tracer-05 binding to C-terminal NanoLuc tagged full length JAK3 (unknown origin) expressed in HEK cells by NanoBRET assayMore data for this Ligand-Target Pair