Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase Mer' and Ligand = 'BDBM497272'
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University of North Carolina at Chapel Hill

US Patent
LigandPNGBDBM497272((1S,4R)-4-(5-([1,4'- bipiperidin]-4-yl)-2-(((S)- p...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47S8SUS Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University of North Carolina at Chapel Hill

US Patent
LigandPNGBDBM497272((1S,4R)-4-(5-([1,4'- bipiperidin]-4-yl)-2-(((S)- p...)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Inhibition of MERTK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90DGJPubMed