Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase SYK' and Ligand = 'BDBM255485'
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Rigel Pharmceuticals, Inc.

US Patent
LigandPNGBDBM255485(US10828301, Compound R926816 | US9499493, R926816)copy SMILEScopy InChI
Affinity DataIC50: 61.5nMAssay Description:Several 2,4-pyrimidinediamine compounds were tested for the ability to inhibit Syk kinase catalyzed phosphorylation of a peptide substrate in a bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47S6WUS Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Rigel Pharmceuticals, Inc.

US Patent
LigandPNGBDBM255485(US10828301, Compound R926816 | US9499493, R926816)copy SMILEScopy InChI
Affinity DataIC50: 61.5nMpH: 7.4 T: 2°CAssay Description:Several 2,4-pyrimidinediamine compounds were tested for the ability to inhibit Syk kinase catalyzed phosphorylation of a peptide substrate in a bioch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WW7GKQUS Patent