Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase receptor UFO' and Ligand = 'BDBM4552'
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Center for Molecular Medicine of the Austrian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Inhibition of AXLMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z15R6PubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Center for Molecular Medicine of the Austrian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of AXL (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M96FSPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Center for Molecular Medicine of the Austrian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of human AXL by scintillation counting method in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M96FSPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Center for Molecular Medicine of the Austrian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077NZPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Center for Molecular Medicine of the Austrian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataKd:  52nMAssay Description:Binding constant for AXL kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8S70PubMed