Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50252659'
TargetUrotensin-2 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50252659((S)-N-(1-(3-bromo-4-(piperidin-4-yloxy)benzyl)pyrr...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [I125]hU2 from human recombinant urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8KTRPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50252659((S)-N-(1-(3-bromo-4-(piperidin-4-yloxy)benzyl)pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of urotensin 2-induced calcium mobiliz...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8KTRPubMed