Found 5 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50459266' 
Affinity DataIC50: 5.60nMAssay Description:Displacement of [Na125I]-synthetic URP from human UT receptor expressed in HEK293 cell membranes incubated for 2 hrs by gamma-countingMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human UT receptor expressed in HEK293 cells co-expressing Gq-polycistronic BRET biosensor assessed as induction of Gq activation ...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as induction of contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Agonist activity at human UT receptor expressed in HEK293 cells co-expressing G12-polycistronic BRET biosensor assessed as induction of G12 activatio...More data for this Ligand-Target Pair
Affinity DataEC50: 182nMAssay Description:Agonist activity at human UT receptor expressed in HEK293 cells co-expressing beta-arrestin1-polycistronic BRET biosensor assessed as induction of be...More data for this Ligand-Target Pair
