Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V1b receptor' and Ligand = 'BDBM50044677'
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ferring Research Institute Inc.

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD426VPubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ferring Research Institute Inc.

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)copy SMILEScopy InChI
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0XXQPubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ferring Research Institute Inc.

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)copy SMILEScopy InChI
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed