TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [3H]-AVP from human V2 receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human V2 receptor expressed in human HeLa cells assessed as inhibition of AVP-induced cAMP accumulation incubated for 10 mins ...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:Agonist activity at human V2 receptor expressed in human HeLa cells assessed as cAMP accumulation incubated for 10 mins by radioimmunoassayMore data for this Ligand-Target Pair
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