Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor' and Ligand = 'BDBM50459404'
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459404(CHEMBL4205046)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-AVP from human V2 receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459404(CHEMBL4205046)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human V2 receptor expressed in human HeLa cells assessed as inhibition of AVP-induced cAMP accumulation incubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg

Curated by ChEMBL
LigandPNGBDBM50459404(CHEMBL4205046)copy SMILEScopy InChI
Affinity DataEC50:  4nMAssay Description:Agonist activity at human V2 receptor expressed in human HeLa cells assessed as cAMP accumulation incubated for 10 mins by radioimmunoassayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed