Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor' and Ligand = 'BDBM85095'
TargetVasopressin V2 receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)copy SMILEScopy InChI
Affinity DataKi:  0.360nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1QW2PubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)copy SMILEScopy InChI
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25T3J1NPubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]AVP from V2 receptor in Wistar rat kidney membranes incubated for 60 mins by microplate scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical Co., Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)copy SMILEScopy InChI
Affinity DataKi:  3.04nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25T3J1NPubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human Vasopressin 2 receptor assessed as inhibition of intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1QW2PubMed