Found 3 Enz. Inhib. hit(s) with Target = 'Vesicular acetylcholine transporter' and Ligand = 'BDBM50378717'
TargetVesicular acetylcholine transporter(Torpedo californica)
Institute of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Institute of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Affinity DataKi: 423nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
Institute of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Institute of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Affinity DataKi: 423nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Rattus norvegicus)
Institute of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Institute of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair