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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'hek293 luciferase' and Ligand = 'BDBM578511'
Target
hek293 luciferase
(Human immunodeficiency virus type 1 group M subtyp...)
TBA
Ligand
BDBM578511
(3-methoxy-5,5- dimethyl-3-(6- methylpyrazin-2- yl)...)
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Affinity Data
EC50: 458nM
Assay Description:
Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2GQ720P
US Patent