Compile Data Set for Download or QSAR
Found 146 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 1277
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283363(N-((6-amino-2,4-dimethylpyridin-3-yl)methyl)- 2-((...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283364(N-((1-aminoisoquinolin-6-yl)methyl)-2-((3- methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283365(N-((3-chloro-6-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283366(N-((6-fluoro-1H-indol-5-yl)methyl)-2-((3- methyl-8...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283367(N-((3-chloro-1H-pyrrolo[2,3-b]pyridin-5- yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283368(N-((5-chloro-1H-indazol-3-yl)methyl)-2-((3- methyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283369(N-((3-chloro-4-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283377(N-((6-amino-4-methylpyridin-3-yl)methyl)-2- ((3-ch...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283379(N-((1-aminoisoquinolin-6-yl)methyl)-2-((3- chloroq...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283381(N-((3-chloro-6-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283382(N-((6-amino-2-methylpyridin-3-yl)methyl)-2- ((3-ch...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283383(N-((6-amino-2,4-dimethylpyridin-3-yl)methyl)- 2-((...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283385(N-((5-chloro-1H-indazol-3-yl)methyl)-2-((3- chloro...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283386(N-((3-chloro-1H-pyrrolo[2,3-b]pyridin-5- yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283382(N-((6-amino-2-methylpyridin-3-yl)methyl)-2- ((3-ch...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283388(N-((3-chloro-4-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283394(N-((6-amino-2,4-dimethylpyridin-3-yl)methyl)- 2-((...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283397(N-((3-chloro-6-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283398(N-((6-amino-2,4-dimethylpyridin-3-yl)methyl)- 2-((...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283399(N-((3-chloro-4-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283400(2-((3-chloro-8-cyanoquinolin-6-yl)methyl)-N- ((6-f...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283402(N-((5-chloro-1H-indazol-3-yl)methyl)-2-((3- chloro...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283403(N-((3-chloro-1H-pyrrolo[2,3-b]pyridin-5- yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283404(N-((6-amino-2-methylpyridin-3-yl)methyl)-2- ((3-ch...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283405(N-((1-aminoisoquinolin-6-yl)methyl)-2-((3- chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283406(6-((4-(((6-amino-2,4-dimethylpyridin-3- yl)methyl)...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283407(3-chloro-6-((4-(((3-chloro-6-fluoro-1H-indol-5- yl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283408(3-chloro-6-((4-(((5-chloro-1H-indazol-3- yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283409(3-chloro-6-((4-(((3-chloro-1H-pyrrolo[2,3- b]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283410(6-((4-(((6-amino-2-methylpyridin-3- yl)methyl)carb...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283411(6-((4-(((6-amino-4-methylpyridin-3- yl)methyl)carb...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283412(6-((4-(((1-aminoisoquinolin-6- yl)methyl)carbamoyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283413(3-chloro-6-((4-(((3-chloro-4-fluoro-1H-indol-5- yl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283414(3-chloro-6-((4-(((6-fluoro-1H-indol-5- yl)methyl)c...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283415(N-((6-amino-2,4-dimethylpyridin-3-yl)methyl)- 2-((...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283416(N-((3-chloro-6-fluoro-1H-indol-5-yl)methyl)-2- ((3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283417(N-((6-amino-2-methylpyridin-3-yl)methyl)-2- ((3-ch...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283418(N-((6-amino-2,4-dimethylpyridin-3-yl)methyl)- 2-((...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283419(N-((1-aminoisoquinolin-6-yl)methyl)-2-((8- cyano-3...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283420(N-((3-chloro-6-fluoro-1H-indol-5-yl)methyl)-2- ((8...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283421(N-((3-chloro-1H-pyrrolo[2,3-b]pyridin-5- yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283422(N-((3-chloro-4-fluoro-1H-indol-5-yl)methyl)-2- ((8...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283423(N-((5-chloro-1H-indazol-3-yl)methyl)-2-((8- cyano-...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283424(2-((8-cyano-3-methylquinolin-6-yl)methyl)-N- ((6-f...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283425(6-((4-(((6-amino-2,4-dimethylpyridin-3- yl)methyl)...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283426(6-((4-(((3-chloro-6-fluoro-1H-indol-5- yl)methyl)c...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283427(6-((4-(((1-aminoisoquinolin-6- yl)methyl)carbamoyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283428(6-((4-(((3-chloro-1H-pyrrolo[2,3-b]pyridin-5- yl)m...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283429(6-((4-(((3-chloro-4-fluoro-1H-indol-5- yl)methyl)c...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
TargetPlasma kallikrein(Homo sapiens (Human))
LIFESCI PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM283430(6-((4-(((5-chloro-1H-indazol-3- yl)methyl)carbamoy...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930W8SUS Patent
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