Compile Data Set for Download or QSAR
Found 50 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 3108
TargetEpidermal growth factor receptor [1-745,751-1210,T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391743(N-(3-((2-((2-methoxy-4-(4-morpholinopiperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391743(N-(3-((2-((2-methoxy-4-(4-morpholinopiperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [1-745,751-1210,T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391742(N-(3-((2-((2-methoxy-4-(1-(methylsulfonyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391733(N-(3-((2-((4-(1-acetyl-1,2,3,6-tetrahydropyridin-4...)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [1-745,751-1210](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391743(N-(3-((2-((2-methoxy-4-(4-morpholinopiperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391731(US10300058, Compound 1 | pyrimidin-4-yl)amino)pyri...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391732(US10300058, Compound 2 | acrylamide )copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391735(N-(6-((2-((4-(1-acetylpiperidin-4-yl)-2-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391736(N-(6-((2-((4-(1-acetyl-1,2,3,6-tetrahydropyridin-4...)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391742(N-(3-((2-((2-methoxy-4-(1-(methylsulfonyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 9.80nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [1-999,L858R](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391743(N-(3-((2-((2-methoxy-4-(4-morpholinopiperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391734(N-(3-((2-((2-acetyl-7-methoxy-1,2,3,4-tetrahydrois...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [1-745,751-1210](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391742(N-(3-((2-((2-methoxy-4-(1-(methylsulfonyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [1-999,L858R](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391742(N-(3-((2-((2-methoxy-4-(1-(methylsulfonyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 88nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 145nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391744(N-(3-((2-((2-methoxy-4-(1-methylpiperidin-4-yl)phe...)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391731(US10300058, Compound 1 | pyrimidin-4-yl)amino)pyri...)copy SMILEScopy InChI
Affinity DataIC50: 323nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391735(N-(6-((2-((4-(1-acetylpiperidin-4-yl)-2-methoxyphe...)copy SMILEScopy InChI
Affinity DataIC50: 423nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391741(US10300058, Compound 26 | pyrimidin-4-yl)amino)phe...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391732(US10300058, Compound 2 | acrylamide )copy SMILEScopy InChI
Affinity DataIC50: 552nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391734(N-(3-((2-((2-acetyl-7-methoxy-1,2,3,4-tetrahydrois...)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391733(N-(3-((2-((4-(1-acetyl-1,2,3,6-tetrahydropyridin-4...)copy SMILEScopy InChI
Affinity DataIC50: 699nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391736(N-(6-((2-((4-(1-acetyl-1,2,3,6-tetrahydropyridin-4...)copy SMILEScopy InChI
Affinity DataIC50: 995nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391743(N-(3-((2-((2-methoxy-4-(4-morpholinopiperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391746(N-(3-((2-((2-methoxy-4-(1-(oxetan-3-yl)piperidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391747(N-(3-((2-((2-methoxy-4-(3-(methylsulfonyl)propoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391739(US10300058, Compound 23 | methyl)pyrimidin-4-yl)am...)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391737(N-(3-((2-((4-(8-acetyl-3,8-diazabicyclo[3.2.1]octa...)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391740(N-(3-((2-((4-(1-(3-fluoropropionyl)piperidin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391742(N-(3-((2-((2-methoxy-4-(1-(methylsulfonyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391745(N-(3-((2-((2-acetyl-1,2,3,4-tetrahydroisoquinoline...)copy SMILEScopy InChI
Affinity DataIC50: 9.90E+3nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391744(N-(3-((2-((2-methoxy-4-(1-methylpiperidin-4-yl)phe...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor [T790M](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391738(N-(3-((2-((2-acetyl-8-methoxy-1,2,3,4-tetrahydrois...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391741(US10300058, Compound 26 | pyrimidin-4-yl)amino)phe...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391743(N-(3-((2-((2-methoxy-4-(4-morpholinopiperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+4nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391746(N-(3-((2-((2-methoxy-4-(1-(oxetan-3-yl)piperidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+4nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 1.53E+5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391747(N-(3-((2-((2-methoxy-4-(3-(methylsulfonyl)propoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391739(US10300058, Compound 23 | methyl)pyrimidin-4-yl)am...)copy SMILEScopy InChI
Affinity DataIC50: 2.94E+5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391737(N-(3-((2-((4-(8-acetyl-3,8-diazabicyclo[3.2.1]octa...)copy SMILEScopy InChI
Affinity DataIC50: 3.32E+5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391740(N-(3-((2-((4-(1-(3-fluoropropionyl)piperidin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 6.83E+5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391742(N-(3-((2-((2-methoxy-4-(1-(methylsulfonyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 8.71E+5nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391745(N-(3-((2-((2-acetyl-1,2,3,4-tetrahydroisoquinoline...)copy SMILEScopy InChI
Affinity DataIC50: 1.28E+6nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84F65US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM391738(N-(3-((2-((2-acetyl-8-methoxy-1,2,3,4-tetrahydrois...)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+6nMAssay Description:Test compounds: a part of compounds of the invention, the chemical names and preparation methods of which can be found in their preparation examples....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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BindingDB Entry DOI: 10.7270/Q2P84F65US Patent