Compile Data Set for Download or QSAR
Found 36 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 41
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101734(US9695160, 31 | US9796707, Compound 31)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101825(US9695160, 39 | US9796707, Compound 39)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM221074(SPHINX31 | US9695160, 12 | US9796707, Compound 12)copy SMILEScopy InChI
Affinity DataIC50: 3.18nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101676(US9695160, 20 | US9796707, Compound 20)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101690(US9695160, 21 | US9796707, Compound 21)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101824(US9695160, 38 | US9796707, Compound 38)copy SMILEScopy InChI
Affinity DataIC50: 5nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101654(US9695160, 14 | US9796707, Compound 14)copy SMILEScopy InChI
Affinity DataIC50: 7.18nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101713(US9695160, 25 | US9796707, Compound 25)copy SMILEScopy InChI
Affinity DataIC50: 14nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101674(US9695160, 19 | US9796707, Compound 19)copy SMILEScopy InChI
Affinity DataIC50: 14nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101671(US9695160, 18 | US9796707, Compound 18)copy SMILEScopy InChI
Affinity DataIC50: 14nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101695(US9695160, 22 | US9796707, Compound 22)copy SMILEScopy InChI
Affinity DataIC50: 15nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101649(US9695160, 13 | US9796707, Compound 13)copy SMILEScopy InChI
Affinity DataIC50: 17nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101657(US9695160, 15 | US9796707, Compound 15)copy SMILEScopy InChI
Affinity DataIC50: 17nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101659(US9695160, 16 | US9796707, Compound 16)copy SMILEScopy InChI
Affinity DataIC50: 38nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM221073(SPHINX scaffold, 3 | US9695160, SPHINX7 | US979670...)copy SMILEScopy InChI
Affinity DataIC50: 55nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101660(US9695160, 17 | US9796707, Compound 17)copy SMILEScopy InChI
Affinity DataIC50: 111nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101832(US9695160, 45 | US9796707, Compound 45)copy SMILEScopy InChI
Affinity DataIC50: 119nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101829(US10696661, Compound 74 | US9695160, 42 | US979670...)copy SMILEScopy InChI
Affinity DataIC50: 164nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101815(US9695160, 36 | US9796707, Compound 36)copy SMILEScopy InChI
Affinity DataIC50: 170nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101830(US9695160, 43 | US9796707, Compound 43)copy SMILEScopy InChI
Affinity DataIC50: 183nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101822(US9695160, 37 | US9796707, Compound 37)copy SMILEScopy InChI
Affinity DataIC50: 323nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101728(US9695160, 30 | US9796707, Compound 30)copy SMILEScopy InChI
Affinity DataIC50: 336nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM221070(SPHINX | US9695160, SPHINX | US9796707, Reference ...)copy SMILEScopy InChI
Affinity DataIC50: 440nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101828(US9695160, 41 | US9796707, Compound 41)copy SMILEScopy InChI
Affinity DataIC50: 493nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101737(US9695160, 32 | US9796707, Compound 32)copy SMILEScopy InChI
Affinity DataIC50: 1.55E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101703(US9695160, 24 | US9796707, Compound 24)copy SMILEScopy InChI
Affinity DataIC50: 3.51E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101696(US9695160, 23 | US9796707, Compound 23)copy SMILEScopy InChI
Affinity DataIC50: 4.01E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101739(US9695160, 33 | US9796707, Compound 33)copy SMILEScopy InChI
Affinity DataIC50: 4.03E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101826(US9695160, 40 | US9796707, Compound 40)copy SMILEScopy InChI
Affinity DataIC50: 4.69E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101740(US9695160, 34 | US9796707, Compound 34)copy SMILEScopy InChI
Affinity DataIC50: 5.31E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101831(US9695160, 44 | US9796707, Compound 44)copy SMILEScopy InChI
Affinity DataIC50: 8.41E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101722(US9695160, 29 | US9796707, Compound 29)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101720(US9695160, 28 | US9796707, Compound 28)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101715(US9695160, 27 | US9796707, Compound 27)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101714(US9695160, 26 | US9796707, Compound 26)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University of Nottingham; NewSouth Innovations PTY Limited

US Patent
LigandPNGBDBM101814(US9695160, 35)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2639MW1US Patent