Compile Data Set for Download or QSAR
Found 131 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 4253
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59116(Hymenialdisine, 27k)copy SMILEScopy InChI
Affinity DataIC50: 10nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59148(Hymenialdisine, 28z)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59146(Hymenialdisine, 28w)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59137(Hymenialdisine, 28p)copy SMILEScopy InChI
Affinity DataIC50: 32nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 37nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59109(Hymenialdisine, 27a)copy SMILEScopy InChI
Affinity DataIC50: 47nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59103(Hymenialdisine, 15)copy SMILEScopy InChI
Affinity DataIC50: 47nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59113(Hymenialdisine, 27g)copy SMILEScopy InChI
Affinity DataIC50: 48nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59140(Hymenialdisine, 28ai)copy SMILEScopy InChI
Affinity DataIC50: 50nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59139(Hymenialdisine, 28aa)copy SMILEScopy InChI
Affinity DataIC50: 50nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59108(Hymenialdisine, 27b)copy SMILEScopy InChI
Affinity DataIC50: 51nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM50256043((Z)-3-bromohymenialdisine | CHEMBL480350 | Hymenia...)copy SMILEScopy InChI
Affinity DataIC50: 51nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59107(Hymenialdisine, 27c)copy SMILEScopy InChI
Affinity DataIC50: 52nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM50256043((Z)-3-bromohymenialdisine | CHEMBL480350 | Hymenia...)copy SMILEScopy InChI
Affinity DataIC50: 56nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59142(Hymenialdisine, 28n)copy SMILEScopy InChI
Affinity DataIC50: 59nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59103(Hymenialdisine, 15)copy SMILEScopy InChI
Affinity DataIC50: 62nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59149(Hymenialdisine, 28v)copy SMILEScopy InChI
Affinity DataIC50: 63nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM50256044(5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...)copy SMILEScopy InChI
Affinity DataIC50: 64nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 70nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 73nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59144(Hymenialdisine, 28ac)copy SMILEScopy InChI
Affinity DataIC50: 75nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59102(Hymenialdisine, 9)copy SMILEScopy InChI
Affinity DataIC50: 79nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59130(Hymenialdisine, 28t)copy SMILEScopy InChI
Affinity DataIC50: 81nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59143(Hymenialdisine, 28ad)copy SMILEScopy InChI
Affinity DataIC50: 81nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59148(Hymenialdisine, 28z)copy SMILEScopy InChI
Affinity DataIC50: 88nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59102(Hymenialdisine, 9)copy SMILEScopy InChI
Affinity DataIC50: 90nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59113(Hymenialdisine, 27g)copy SMILEScopy InChI
Affinity DataIC50: 109nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 111nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 112nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59136(Hymenialdisine, 28ah)copy SMILEScopy InChI
Affinity DataIC50: 118nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59110(Hymenialdisine, 27e)copy SMILEScopy InChI
Affinity DataIC50: 120nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59131(Hymenialdisine, 28g)copy SMILEScopy InChI
Affinity DataIC50: 125nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59139(Hymenialdisine, 28aa)copy SMILEScopy InChI
Affinity DataIC50: 147nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59114(Hymenialdisine, 27i)copy SMILEScopy InChI
Affinity DataIC50: 163nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59130(Hymenialdisine, 28t)copy SMILEScopy InChI
Affinity DataIC50: 171nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59115(Hymenialdisine, 27j)copy SMILEScopy InChI
Affinity DataIC50: 175nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59150(Hymenialdisine, 28ae)copy SMILEScopy InChI
Affinity DataIC50: 177nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM50256044(5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...)copy SMILEScopy InChI
Affinity DataIC50: 177nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59107(Hymenialdisine, 27c)copy SMILEScopy InChI
Affinity DataIC50: 177nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59134(Hymenialdisine, 28ab)copy SMILEScopy InChI
Affinity DataIC50: 179nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59114(Hymenialdisine, 27i)copy SMILEScopy InChI
Affinity DataIC50: 187nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59108(Hymenialdisine, 27b)copy SMILEScopy InChI
Affinity DataIC50: 191nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59109(Hymenialdisine, 27a)copy SMILEScopy InChI
Affinity DataIC50: 213nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59103(Hymenialdisine, 15)copy SMILEScopy InChI
Affinity DataIC50: 220nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 250nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59104(Hymenialdisine, 18)copy SMILEScopy InChI
Affinity DataIC50: 251nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59104(Hymenialdisine, 18)copy SMILEScopy InChI
Affinity DataIC50: 268nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59105(Hymenialdisine, 16)copy SMILEScopy InChI
Affinity DataIC50: 363nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59131(Hymenialdisine, 28g)copy SMILEScopy InChI
Affinity DataIC50: 399nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute of the Novartis Research Foundation

LigandPNGBDBM59112(Hymenialdisine, 27h)copy SMILEScopy InChI
Affinity DataIC50: 400nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN14M9PubMed
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