Compile Data Set for Download or QSAR
Found 16 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50000004
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239077(CHEMBL4082302)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239089(CHEMBL4098261)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:In vitro binding to human erythrocyte Carbonic anhydrase II was determined by fluorescence competition assay employing the fluorescent CA inhibitor d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239081(CHEMBL4081347)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239078(CHEMBL4062127)copy SMILEScopy InChI
Affinity DataKi:  230nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239074(CHEMBL4071224)copy SMILEScopy InChI
Affinity DataKi:  270nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239080(CHEMBL4097869)copy SMILEScopy InChI
Affinity DataKi:  410nMAssay Description:Compound was tested for its inhibition activity against the 5-LO in isolated enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)copy SMILEScopy InChI
Affinity DataKi:  420nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239079(CHEMBL4070752)copy SMILEScopy InChI
Affinity DataKi:  470nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239075(CHEMBL4067010)copy SMILEScopy InChI
Affinity DataKi:  730nMAssay Description:In vitro binding to human erythrocyte Carbonic anhydrase II was determined by fluorescence competition assay employing the fluorescent CA inhibitor d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239086(CHEMBL4105602)copy SMILEScopy InChI
Affinity DataKi:  760nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239088(CHEMBL4094488)copy SMILEScopy InChI
Affinity DataKi:  810nMAssay Description:In vitro binding to human erythrocyte Carbonic anhydrase II was determined by fluorescence competition assay employing the fluorescent CA inhibitor d...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239076(CHEMBL4100319)copy SMILEScopy InChI
Affinity DataKi:  850nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239084(CHEMBL4088240)copy SMILEScopy InChI
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239085(CHEMBL4094073)copy SMILEScopy InChI
Affinity DataKi:  1.19E+3nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239082(CHEMBL4073436)copy SMILEScopy InChI
Affinity DataKi:  1.24E+3nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50239087(CHEMBL4090152)copy SMILEScopy InChI
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of 6-carboxyfluorescein succinimidyl ester fluorescence tagged-Bid BH3 peptide (79 to 99 residues) binding to Bcl-2 (unknown origin) after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6SMCPubMed