Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50001342
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78HRZPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276840(CHEMBL4160471)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78HRZPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276841(CHEMBL4161963)copy SMILEScopy InChI
Affinity DataIC50: 447nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78HRZPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276839(CHEMBL4170184)copy SMILEScopy InChI
Affinity DataIC50: 891nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78HRZPubMed