Compile Data Set for Download or QSAR
Found 23 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50001424
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50267750(CHEMBL1078685)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279097(CHEMBL4160962)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279093(CHEMBL4171577)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279092(CHEMBL4172836)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279091(CHEMBL4164929)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279055(CHEMBL4176624)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279094(CHEMBL4164363)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279062(CHEMBL4166015)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279056(CHEMBL4167511)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279078(CHEMBL4168690)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279053(CHEMBL4159596)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of bovine xanthine oxidase assessed as reduction in uric acid formation using xanthine as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279052(CHEMBL4165271)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of bovine xanthine oxidase assessed as reduction in uric acid formation using xanthine as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279079(CHEMBL4173175)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279077(CHEMBL4176545)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279054(CHEMBL4159940)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of bovine xanthine oxidase assessed as reduction in uric acid formation using xanthine as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279090(CHEMBL4161510)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279076(CHEMBL4162571)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279089(CHEMBL4173257)copy SMILEScopy InChI
Affinity DataIC50: 9.50E+3nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279088(CHEMBL4170588)copy SMILEScopy InChI
Affinity DataIC50: 1.92E+4nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279111(CHEMBL4169071)copy SMILEScopy InChI
Affinity DataIC50: 2.26E+4nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279096(CHEMBL4165035)copy SMILEScopy InChI
Affinity DataIC50: 3.28E+4nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
China Medical University

Curated by ChEMBL
LigandPNGBDBM50279095(CHEMBL4160555)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+4nMAssay Description:Antagonistic activity against the P2X7 ion channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K90PubMed