Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50001929
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50450580(CHEMBL4169884)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of human Nav1.5 expressed in HEK293 cells at holding potential of -20 mV after 10 mins by patchxpress-based electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4ZB0PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50450593(CHEMBL4164272)copy SMILEScopy InChI
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human Nav1.5 expressed in HEK293 cells at holding potential of -20 mV after 10 mins by patchxpress-based electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4ZB0PubMed
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50450581(CHEMBL4159169)copy SMILEScopy InChI
Affinity DataIC50: 6.64E+3nMAssay Description:Inhibition of human Nav1.5 expressed in HEK293 cells at holding potential of -20 mV after 10 mins by patchxpress-based electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4ZB0PubMed