Compile Data Set for Download or QSAR
Found 25 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50008271
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517275(CHEMBL4469040)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517268(CHEMBL4475144)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM109086(US10793535, Cmpd ID 727 | US8604016, 670 | US99382...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517258(CHEMBL4462204)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517276(CHEMBL4474779)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517261(CHEMBL4474767)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517270(CHEMBL4451104)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517265(CHEMBL4566474)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517263(CHEMBL4442957)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50400050(CHEMBL2177757 | US10793535, Cmpd ID 1 | US11191732...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM108625(US8604016, 200 | US9938267, Cmpd ID 200)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517267(CHEMBL4590724)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517260(CHEMBL4441674)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517272(CHEMBL4522431)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517266(CHEMBL4441375)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517262(CHEMBL4593057)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517264(CHEMBL4582249)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM108460(CHEMBL2178393 | US11191732, Example 1 | US8604016,...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517273(CHEMBL4459382)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517274(CHEMBL4436915)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50400072(CHEMBL2178396 | US11191732, Example 3)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517271(CHEMBL4565066)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517269(CHEMBL4550553)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM108464(US8604016, 21 | US9938267, Cmpd ID 21)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50517259(CHEMBL4465855)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FF2PubMed