Compile Data Set for Download or QSAR
Found 12 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50009072
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525156(CHEMBL4476248)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525162(CHEMBL4434651)copy SMILEScopy InChI
Affinity DataKi:  880nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525160(CHEMBL4522230)copy SMILEScopy InChI
Affinity DataKi:  990nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525157(CHEMBL4460155)copy SMILEScopy InChI
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525158(CHEMBL4515564)copy SMILEScopy InChI
Affinity DataKi:  1.23E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525159(CHEMBL4471293)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525161(CHEMBL4557901)copy SMILEScopy InChI
Affinity DataKi:  1.44E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525154(CHEMBL4581547)copy SMILEScopy InChI
Affinity DataKi:  1.72E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525163(CHEMBL4566271)copy SMILEScopy InChI
Affinity DataKi:  2.03E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50525162(CHEMBL4434651)copy SMILEScopy InChI
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BGPPubMed