Compile Data Set for Download or QSAR
Found 57 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50012933
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124496(CHEMBL368996 | Pyrazin-2-yl-carbamic acid 4-[6-(5-...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124459(Butyl-carbamic acid 4-[6-(5-isopropyl-pyridine-2-s...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124470(CHEMBL264035 | Phenyl-carbamic acid 4-[6-(5-isopro...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124485(CHEMBL367036 | Phenyl-carbamic acid 4-[6-(5-isopro...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124474(CHEMBL94786 | Pyridin-2-yl-carbamic acid 4-[6-(5-i...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124461(4-tert-Butyl-N-[6-(4-hydroxy-but-2-ynyloxy)-5-(2-m...)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124504(5-Isopropyl-pyridine-2-sulfonic acid [6-(4-hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124480(4-tert-Butyl-N-[6-(4-hydroxy-but-2-ynyloxy)-5-(2-m...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124483(5-Isopropyl-pyridine-2-sulfonic acid [6-(4-hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124473(4-tert-Butyl-N-[2-(2-hydroxymethyl-pyridin-4-yl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124498(CHEMBL368386 | Pyridin-2-yl-carbamic acid 4-[6-(5-...)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124490(5-Isopropyl-pyridine-2-sulfonic acid [6-(4-hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 183nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124465(CHEMBL367453 | Pyridin-2-yl-carbamic acid 4-[5-(2-...)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124467(CHEMBL139734 | N-[6-(4-Benzyloxy-but-2-ynyloxy)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 199nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124493(5-Isopropyl-pyridine-2-sulfonic acid [2-(2-hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 205nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124452(Butyl-carbamic acid 4-[5-(2-methoxy-phenoxy)-6-(5-...)copy SMILEScopy InChI
Affinity DataIC50: 207nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124476(5-Isopropyl-pyridine-2-sulfonic acid {5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 221nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124492(CHEMBL275897 | Pyrazin-2-yl-carbamic acid 4-[6-(5-...)copy SMILEScopy InChI
Affinity DataIC50: 236nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124454(4-tert-Butyl-N-{5-(2-methoxy-phenoxy)-2-[2-(5-oxo-...)copy SMILEScopy InChI
Affinity DataIC50: 238nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124453(CHEMBL175058 | Pyrazin-2-yl-carbamic acid 4-[5-(2-...)copy SMILEScopy InChI
Affinity DataIC50: 241nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124506(4-tert-Butyl-N-{5-(2-methoxy-phenoxy)-6-prop-2-yny...)copy SMILEScopy InChI
Affinity DataIC50: 258nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50061101(4-(1,1-Dimethylethyl)-N-(6-(2-hydroxyethoxy)-5-(2-...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124486(5-Isopropyl-pyridine-2-sulfonic acid {5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 294nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124479(4-tert-Butyl-N-[5-(2-methoxy-phenoxy)-6-prop-2-yny...)copy SMILEScopy InChI
Affinity DataIC50: 295nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124482(5-Isopropyl-pyridine-2-sulfonic acid {5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 366nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124503(CHEMBL163638 | Phenyl-carbamic acid 4-[5-(2-methox...)copy SMILEScopy InChI
Affinity DataIC50: 589nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124469(CHEMBL175278 | Cyclohexyl-carbamic acid 4-[5-(2-me...)copy SMILEScopy InChI
Affinity DataIC50: 603nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124463(5-Methyl-pyridine-2-sulfonic acid [6-(4-hydroxy-bu...)copy SMILEScopy InChI
Affinity DataIC50: 612nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124495(CHEMBL366885 | Pyridin-4-yl-carbamic acid 4-[5-(2-...)copy SMILEScopy InChI
Affinity DataIC50: 656nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124455(4-tert-Butyl-N-[6-(4-hydroxy-but-2-ynyloxy)-5-(2-m...)copy SMILEScopy InChI
Affinity DataIC50: 744nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124475(5-Isopropyl-pyridine-2-sulfonic acid [5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 746nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124464(5-Isopropyl-pyridine-2-sulfonic acid [5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 823nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124471(4-tert-Butyl-N-[6-(4-hydroxy-but-2-ynyloxy)-5-(2-m...)copy SMILEScopy InChI
Affinity DataIC50: 832nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124477(4-tert-Butyl-N-[5-(2-methoxy-phenoxy)-6-prop-2-yny...)copy SMILEScopy InChI
Affinity DataIC50: 903nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124456(CHEMBL176741 | Pyridin-3-yl-carbamic acid 4-[5-(2-...)copy SMILEScopy InChI
Affinity DataIC50: 920nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124460(4-tert-Butyl-N-[5-(2-methoxy-phenoxy)-6-(4-phenoxy...)copy SMILEScopy InChI
Affinity DataIC50: 973nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124481(5-Methyl-pyridine-2-sulfonic acid [2-(2-hydroxymet...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124487(5-Methyl-pyridine-2-sulfonic acid {5-(2-methoxy-ph...)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124500(CHEMBL368860 | Pyridin-2-yl-carbamic acid 4-[6-(4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124462(4-tert-Butyl-N-[6-(4-methoxy-but-2-ynyloxy)-5-(2-m...)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124497(4-tert-Butyl-N-[5-(2-methoxy-phenoxy)-6-prop-2-yny...)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124458(CHEMBL367767 | Pyrazin-2-yl-carbamic acid 4-[6-(4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124466(5-Methyl-pyridine-2-sulfonic acid [6-(4-hydroxy-bu...)copy SMILEScopy InChI
Affinity DataIC50: 1.52E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124507(5-Methyl-pyridine-2-sulfonic acid {5-(2-methoxy-ph...)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124505(5-Isopropyl-pyridine-2-sulfonic acid [5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 1.95E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124457(5-Isopropyl-pyridine-2-sulfonic acid [6-(4-hydroxy...)copy SMILEScopy InChI
Affinity DataIC50: 2.03E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124484(CHEMBL367339 | N-[6-Allyloxy-5-(2-methoxy-phenoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 2.09E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124488(4-tert-Butyl-N-[5-(2-methoxy-phenoxy)-6-pent-2-yny...)copy SMILEScopy InChI
Affinity DataIC50: 2.28E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124494(5-Methyl-pyridine-2-sulfonic acid {5-(2-methoxy-ph...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals Ltd

Curated by ChEMBL
LigandPNGBDBM50124501(5-Isopropyl-pyridine-2-sulfonic acid [5-(2-methoxy...)copy SMILEScopy InChI
Affinity DataIC50: 2.62E+3nMAssay Description:In vitro inhibitory concentration required against [125I]-ET-1 binding to membranes of CHO cells expressing human ETB receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28C9VK8PubMed
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