Compile Data Set for Download or QSAR
Found 28 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50014936
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581295(CHEMBL5081077)copy SMILES
Affinity DataEC50:  0.813nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataEC50: >0.0501nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581297(CHEMBL5091236)copy SMILES
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50263842(CHEMBL4099889)copy SMILEScopy InChI
Affinity DataEC50:  65nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581298(CHEMBL5094168)copy SMILES
Affinity DataEC50:  0.0832nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581299(CHEMBL5075506)copy SMILES
Affinity DataEC50:  0.141nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581300(CHEMBL5091245)copy SMILES
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581301(CHEMBL5093939)copy SMILES
Affinity DataEC50:  0.759nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581302(CHEMBL5075712)copy SMILES
Affinity DataEC50:  0.138nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581303(CHEMBL5087859)copy SMILES
Affinity DataEC50: >0.0501nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581304(CHEMBL5077811)copy SMILES
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581305(CHEMBL5085972)copy SMILES
Affinity DataEC50:  8.70nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581306(CHEMBL5077095)copy SMILES
Affinity DataEC50:  0.135nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581307(CHEMBL5090670)copy SMILES
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581308(CHEMBL5090285)copy SMILES
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581309(CHEMBL5078687)copy SMILES
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581310(CHEMBL5077144)copy SMILES
Affinity DataEC50:  0.427nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581311(CHEMBL5083551)copy SMILES
Affinity DataEC50:  0.0562nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581312(CHEMBL5094215)copy SMILES
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581313(CHEMBL5087839)copy SMILES
Affinity DataEC50: <0.0501nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581314(CHEMBL5090946)copy SMILES
Affinity DataEC50:  0.0912nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581315(CHEMBL5080489)copy SMILES
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581316(CHEMBL5080784)copy SMILES
Affinity DataEC50:  0.692nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581317(CHEMBL5087814)copy SMILES
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581318(CHEMBL5076315)copy SMILES
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581319(BIM-22493 | RM-493 | SETMELANOTIDE | Setmelanotide)copy SMILES
Affinity DataEC50:  0.158nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50389769(BREMELANOTIDE)copy SMILEScopy InChI
Affinity DataEC50:  0.0776nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50581296(CHEMBL5092761)copy SMILES
Affinity DataEC50:  0.0646nMAssay Description:Agonist activity at human melanocortin receptor 1 expressed in human T-Rex-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed