Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50016436
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM50168964((3S,4aR,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenylamin...)copy SMILEScopy InChI
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM50168965((3S,4aS,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenoxy]-d...)copy SMILEScopy InChI
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)copy SMILEScopy InChI
Affinity DataKi:  4.16E+3nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM50168963((3S,4aS,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenoxy]-d...)copy SMILEScopy InChI
Affinity DataKi:  7.37E+3nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM50207594(2,3-Dihydroxy-6-nitro-benzo[f]quinoxaline-7-sulfon...)copy SMILEScopy InChI
Affinity DataKi:  1.17E+4nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM50168962((3S,4aR,6S,8aR)-6-(4-Carboxy-benzyl)-decahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  1.71E+4nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro de Investigación Lilly

Curated by ChEMBL
LigandPNGBDBM50168966((3S,4aR,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenylamin...)copy SMILEScopy InChI
Affinity DataKi:  3.18E+4nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ3ZDMPubMed