Compile Data Set for Download or QSAR
Found 23 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50018524
LigandPNGBDBM370147(US10233188, Example 36 | US10800783, Example 36 | ...)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM467013((-)-6-(2,2-difluoroethyl)-8-[(1R*,2R*)-2-hydroxy-2...)copy SMILEScopy InChI
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370205(US10233188, Example 92 | US10800783, Example 92 | ...)copy SMILEScopy InChI
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370121(6-(difluoromethyl)-8-[(1R,2R)-2-hydroxy-2-methylcy...)copy SMILEScopy InChI
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM370120(6-chloro-8-[(1R,2R)-2-hydroxy-2-methylcyclopentyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370113(8-[(1R,2R)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(m...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370130(US10233188, Example 19 | US10800783, Example 19 | ...)copy SMILEScopy InChI
Affinity DataKi:  0.360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370133(US10233188, Example 22 | US10800783, Example 22 | ...)copy SMILEScopy InChI
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370112(8-cyclopentyl-2-{[1-(methylsulfonyl)piperidin-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50609168(CHEMBL5277190)copy SMILES
Affinity DataKi:  0.880nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370248((8-cyclopentyl-2-{[1-(methylsulfonyl)piperidin-4-y...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370140(US10233188, Example 29 | US10800783, Example 29 | ...)copy SMILEScopy InChI
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370258(BDBM467153 | US10233188, Example 145)copy SMILES
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50609168(CHEMBL5277190)copy SMILES
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM370257(BDBM467152 | US10233188, Example 144)copy SMILES
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM370256(BDBM467151 | US10233188, Example 143)copy SMILES
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM370277(BDBM467172 | US10233188, Example 164)copy SMILES
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50609167(CHEMBL5283828)copy SMILES
Affinity DataKi:  4.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50609166(CHEMBL5280928)copy SMILES
Affinity DataKi:  5.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50609170(CHEMBL5266837)copy SMILES
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50609171(CHEMBL5288078)copy SMILES
Affinity DataKi:  82nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50609169(CHEMBL5275378)copy SMILES
Affinity DataKi:  1.36E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM6309(6-Acetyl-8-cyclopentyl-5-methyl-2-(5-piperazin-1-y...)copy SMILEScopy InChI
Affinity DataKi: >2.66E+3nMMore data for this Ligand-Target Pair
In DepthDetails